Sharpless, K Barry

Publication with MATCHING institution:

Dong J, Sharpless KB, Kwisnek L, Oakdale JS (2014) SuFEx-based synthesis of polysulfates. Angewandte Chemie -
International Edition. [IF=2.456, Cited=67, 25100330].
Sharpless KB, Finn MG, Martín VS (2015) Tsutomu Katsuki (1946-2014). Angewandte Chemie - International Edition.
[IF=2.456, Cited=0, 25766459].
Chen W, Dong J, Li S, ..., Kelly JW (2015) Synthesis of Sulfotyrosine-Containing Peptides by Incorporating
Fluorosulfated Tyrosine Using an Fmoc-Based Solid-Phase Strategy. Angewandte Chemie - International Edition. [IF=2.456,
Cited=20, 26696445].
Qin HL, Zheng Q, Bare GAL, ..., Sharpless KB (2016) A Heck-Matsuda Process for the Synthesis of β-Arylethenesulfonyl
Fluorides: Selectively Addressable Bis-electrophiles for SuFEx Click Chemistry. Angewandte Chemie - International
Edition. [IF=2.456, Cited=42, 27723200].
Li S, Wu P, Moses JE, Sharpless KB (2017) Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride
Exchange Connections of Diverse Modules Launched From An SOF₄ Hub. Angewandte Chemie - International Edition.
[IF=2.456, Cited=44, 28165188].
Wang H, Zhou F, Ren G, ..., Wu P (2017) SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts.
Angewandte Chemie - International Edition. [IF=2.456, Cited=37, 28792119].
Zha GF, Zheng Q, Leng J, ..., Sharpless KB (2017) Palladium-Catalyzed Fluorosulfonylvinylation of Organic Iodides.
Angewandte Chemie - International Edition. [IF=2.456, Cited=24, 28370917].
Gao B, Li S, Wu P, ..., Sharpless KB (2018) SuFEx Chemistry of Thionyl Tetrafluoride (SOF₄ ) with
Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides, and Sulfonimidates.
Angewandte Chemie - International Edition. [IF=2.456, Cited=30, 29314580].
Smedley CJ, Zheng Q, Gao B, ..., Moses JE (2019) Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl
Fluorides and Iminosulfur Oxydifluorides. Angewandte Chemie - International Edition. [IF=2.456, Cited=18, 30740848].
Liu F, Wang H, Li S, ..., Sharpless KB (2019) Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride
(SOF₄ )-Derived Connective Hubs for Bioconjugation to DNA and Proteins. Angewandte Chemie - International
Edition. [IF=2.456, Cited=37, 30998840].
Smedley CJ, Li G, Barrow AS, ..., Moses JE (2020) Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable
Pharmacophores from 2-Substituted-Alkynyl-1-Sulfonyl Fluoride (SASF) Hubs. Angewandte Chemie - International Edition.
[IF=2.456, Cited=21, 32301265].
Sun S, Gao B, Chen J, ..., Dong J (2021) Fluorosulfuryl Isocyanate Enabled SuFEx Ligation of Alcohols and Amines.
Angewandte Chemie - International Edition. [IF=2.456, Cited=4, 34259368].
Zhang E, Tang J, Li S, ..., Sharpless KB (2016) Chemoselective Synthesis of Polysubstituted Pyridines from Heteroaryl
Fluorosulfates. Chemistry - A European Journal. [IF=0.899, Cited=15, 26990693].
Silverman SM, Moses JE, Sharpless KB (2016) Reengineering Antibiotics to Combat Bacterial Resistance: Click Chemistry
[1,2,3]-Triazole Vancomycin Dimers with Potent Activity against MRSA and VRE. Chemistry - A European Journal. [IF=0.899,
Cited=23, 27747932].
Gahtory D, Sen R, Pujari S, ..., Zuilhof H (2018) Quantitative and Orthogonal Formation and Reactivity of SuFEx
Platforms. Chemistry - A European Journal. [IF=0.899, Cited=15, 29949211].
Kovarik Z, Kalisiak J, Hrvat NM, ..., Taylor P (2019) Reversal of Tabun Toxicity Enabled by a Triazole-Annulated Oxime
Library-Reactivators of Acetylcholinesterase. Chemistry - A European Journal. [IF=0.899, Cited=6, 30458057].
Yang Y, Chen M, Wu M, ..., Wu P (2023) Chemoenzymatic Tagging of Tn/TF/STF Antigens in Living Systems. Israel Journal of
Chemistry. [IF=0.673, Cited=0, 38737670].
Taylor P, Yan-Jye S, Momper J, ..., Sharpless KB (2019) Assessment of ionizable, zwitterionic oximes as reactivating
antidotal agents for organophosphate exposure. None. [IF=None, Cited=10, 31100277].
McFadden WM, Casey-Moore MC, Bare GAL, ..., Sarafianos SG (2024) Identification of clickable HIV-1 capsid-targeting
probes for viral replication inhibition. Cell Chemical Biology. [IF=1.446, Cited=0, 38518746].
Sun S, Homer JA, Smedley CJ, ..., Moses JE (2023) Phosphorus fluoride exchange: Multidimensional catalytic click
chemistry from phosphorus connective hubs. Chem. [IF=2.863, Cited=0, 38882554].
Li H, Chang BS, Kim H, ..., Liu Y (2023) High-performing polysulfate dielectrics for electrostatic energy storage under
harsh conditions. Joule. [IF=4.95, Cited=6, 37034575].
Kovarik Z, Maček Hrvat N, Kalisiak J, ..., Taylor P (2019) Counteracting tabun inhibition by reactivation by pyridinium
aldoximes that interact with active center gorge mutants of acetylcholinesterase. Toxicology and Applied Pharmacology.
[IF=0.883, Cited=2, 30978400].
Maček Hrvat N, Kalisiak J, Šinko G, ..., Kovarik Z (2019) Evaluation of high-affinity phenyltetrahydroisoquinoline
aldoximes, linked through anti-triazoles, as reactivators of phosphylated cholinesterases. Toxicology Letters.
[IF=0.908, Cited=7, 31863869].
Zheng Q, Dong J, Sharpless KB (2016) Ethenesulfonyl Fluoride (ESF): An On-Water Procedure for the Kilogram-Scale
Preparation. Journal of Organic Chemistry. [IF=0.885, Cited=26, 27764941].
Liang Q, Xing P, Huang Z, ..., Jiang B (2015) Palladium-catalyzed, ligand-free Suzuki reaction in water using aryl
fluorosulfates. Organic Letters. [IF=1.091, Cited=27, 25856416].
Garnar-Wortzel L, Bishop TR, Kitamura S, ..., Erb MA (2021) Chemical Inhibition of ENL/AF9 YEATS Domains in Acute
Leukemia. ACS Central Science. [IF=2.363, Cited=29, 34079898].
Kim H, Zhao J, Bae J, ..., Wu P (2021) Chain-Growth Sulfur(VI) Fluoride Exchange Polycondensation: Molecular Weight
Control and Synthesis of Degradable Polysulfates. ACS Central Science. [IF=2.363, Cited=5, 34841062].
Morris GM, Green LG, Radić Z, ..., Grynszpan F (2013) Automated docking with protein flexibility in the design of
femtomolar "click chemistry" inhibitors of acetylcholinesterase. Journal of Chemical Information and Modeling.
[IF=1.379, Cited=14, 23451944].
Himo F, Demko ZP, Noodleman L, Sharpless KB (2002) Mechanisms of tetrazole formation by addition of azide to nitriles.
Journal of the American Chemical Society. [IF=2.573, Cited=56, 12371861].
Wang Q, Chan TR, Hilgraf R, ..., Finn MG (2003) Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2]
cycloaddition. Journal of the American Chemical Society. [IF=2.573, Cited=605, 12630856].
Himo F, Demko ZP, Noodleman L, Sharpless KB (2003) Why is tetrazole formation by addition of azide to organic nitriles
catalyzed by zinc(II) salts? Journal of the American Chemical Society. [IF=2.573, Cited=56, 12914461].
Lee LV, Mitchell ML, Huang SJ, ..., Wong CH (2003) A potent and highly selective inhibitor of human
alpha-1,3-fucosyltransferase via click chemistry. Journal of the American Chemical Society. [IF=2.573, Cited=148, 12904015].
Krasiński A, Radić Z, Manetsch R, ..., Sharpless KB (2005) In situ selection of lead compounds by click chemistry:
target-guided optimization of acetylcholinesterase inhibitors. Journal of the American Chemical Society. [IF=2.573,
Cited=120, 15869290].
Manetsch R, Krasiński A, Radić Z, ..., Sharpless KB (2004) In situ click chemistry: enzyme inhibitors made to their own
specifications. Journal of the American Chemical Society. [IF=2.573, Cited=144, 15469276].
Himo F, Lovell T, Hilgraf R, ..., Sharpless KB (2005) Copper(I)-catalyzed synthesis of azoles. DFT study predicts
unprecedented reactivity and intermediates. Journal of the American Chemical Society. [IF=2.573, Cited=410, 15631470].
Feldman AK, Colasson B, Sharpless KB (2005) The allylic azide rearrangement: achieving selectivity. Journal of the
American Chemical Society. [IF=2.573, Cited=41, 16190677].
Zhang L, Chen X, Xue P, ..., Jia G (2005) Ruthenium-catalyzed cycloaddition of alkynes and organic azides. Journal of
the American Chemical Society. [IF=2.573, Cited=287, 16287266].
Millward SW, Henning RK, Kwong GA, ..., Sharpless KB (2011) Iterative in situ click chemistry assembles a branched
capture agent and allosteric inhibitor for Akt1. Journal of the American Chemical Society. [IF=2.573, Cited=22, 21962254].
Grimster NP, Stump B, Fotsing JR, ..., Taylor P (2012) Generation of candidate ligands for nicotinic acetylcholine
receptors via in situ click chemistry with a soluble acetylcholine binding protein template. Journal of the American
Chemical Society. [IF=2.573, Cited=29, 22394239].
Grimster NP, Connelly S, Baranczak A, ..., Kelly JW (2013) Aromatic sulfonyl fluorides covalently kinetically stabilize
transthyretin to prevent amyloidogenesis while affording a fluorescent conjugate. Journal of the American Chemical
Society. [IF=2.573, Cited=66, 23350654].
Kalisiak J, Trauger SA, Kalisiak E, ..., Siuzdak G (2009) Identification of a new endogenous metabolite and the
characterization of its protein interactions through an immobilization approach. Journal of the American Chemical
Society. [IF=2.573, Cited=26, 19055353].
Zheng Q, Xu H, Wang H, ..., Wu P (2021) Sulfur [¹⁸F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-
Stage Radiosynthesis. Journal of the American Chemical Society. [IF=2.573, Cited=37, 33630577].
Baranczak A, Liu Y, Connelly S, ..., Kelly JW (2015) A fluorogenic aryl fluorosulfate for intraorganellar transthyretin
imaging in living cells and in Caenorhabditis elegans. Journal of the American Chemical Society. [IF=2.573, Cited=33, 26051248].
Bourne Y, Sharpless KB, Taylor P, Marchot P (2016) Steric and Dynamic Parameters Influencing In Situ Cycloadditions to
Form Triazole Inhibitors with Crystalline Acetylcholinesterase. Journal of the American Chemical Society. [IF=2.573,
Cited=18, 26731630].
Chen W, Dong J, Plate L, ..., Kelly JW (2016) Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s)
through Chemoselective SuFEx Reaction with a Binding Site Tyr Residue. Journal of the American Chemical Society.
[IF=2.573, Cited=97, 27191344].
Mortenson DE, Brighty GJ, Plate L, ..., Kelly JW (2017) "Inverse Drug Discovery" Strategy To Identify Proteins That Are
Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates. Journal of the American Chemical Society.
[IF=2.573, Cited=91, 29265822].
Liu Z, Li J, Li S, ..., Wu P (2018) SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization. Journal of the
American Chemical Society. [IF=2.573, Cited=69, 29451783].
Johnson SM, Petrassi HM, Palaninathan SK, ..., Kelly JW (2005) Bisaryloxime ethers as potent inhibitors of transthyretin
amyloid fibril formation. Journal of Medicinal Chemistry. [IF=1.655, Cited=42, 15743199].
Whiting M, Tripp JC, Lin YC, ..., Sharpless KB (2006) Rapid discovery and structure-activity profiling of novel
inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of
1,2,3-triazoles and their further functionalization. Journal of Medicinal Chemistry. [IF=1.655, Cited=62, 17181152].
Sit RK, Amitai G, Sharpless KB, ..., Radić Z (2014) Imidazole aldoximes effective in assisting butyrylcholinesterase
catalysis of organophosphate detoxification. Journal of Medicinal Chemistry. [IF=1.655, Cited=35, 24571195].
Valdez CA, Tripp JC, Miyamoto Y, ..., Eckmann L (2009) Synthesis and electrochemistry of 2-ethenyl and 2-ethanyl
derivatives of 5-nitroimidazole and antimicrobial activity against Giardia lamblia. Journal of Medicinal Chemistry.
[IF=1.655, Cited=32, 19480409].
Marzinzik AL, Sharpless KB (2001) A simple method for the preparation of N-sulfonylsulfilimines from sulfides. Journal
of Organic Chemistry. [IF=0.885, Cited=16, 11429835].
Demko ZP, Sharpless KB (2001) Preparation of 5-substituted 1H-tetrazoles from nitriles in water. Journal of Organic
Chemistry. [IF=0.885, Cited=147, 11722189].
Converso A, Burow K, Marzinzik A, ..., Finn MG (2001) 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: a privileged, bivalent
scaffold for the display of nucleophilic components. Journal of Organic Chemistry. [IF=0.885, Cited=5, 11397181].
Converso A, Saaidi PL, Sharpless KB, Finn MG (2004) Nucleophilic substitution by grignard reagents on sulfur mustards.
Journal of Organic Chemistry. [IF=0.885, Cited=4, 15471488].
Yoo EJ, Ahlquist M, Bae I, ..., Chang S (2008) Mechanistic studies on the Cu-catalyzed three-component reactions of
sulfonyl azides, 1-alkynes and amines, alcohols, or water: dichotomy via a common pathway. Journal of Organic Chemistry.
[IF=0.885, Cited=52, 18557650].
Chang HT, Sharpless KB (1996) Molar Scale Synthesis of Enantiopure Stilbene Oxide. Journal of Organic Chemistry.
[IF=0.885, Cited=4, 11667495].
Sharpless KB (1996) Ligand-Dependent Reversal of Facial Selectivity in the Asymmetric Dihydroxylation. Journal of
Organic Chemistry. [IF=0.885, Cited=10, 11667767].
Gypser A, Michel D, Sharpless KB (1998) Dihydroxylation of Polyenes Using Narasaka's Modification of the Upjohn
Procedure. Journal of Organic Chemistry. [IF=0.885, Cited=8, 11672379].
Sharpless KB (1999) The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates. Journal of Organic
Chemistry. [IF=0.885, Cited=18, 11674762].
Weide T, Saldanha SA, Minond D, ..., Hodder PS (2010) NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-
Lactamase: Synthesis and Structure-Activity Studies. ACS Medicinal Chemistry Letters. [IF=0.873, Cited=31, 20625539].
Demko ZP, Bartsch M, Sharpless KB (2000) Primary amides. A general nitrogen source for catalytic asymmetric
aminohydroxylation of olefins. Organic Letters. [IF=1.091, Cited=7, 10930248].
Chuang TH, Sharpless KB (2000) Applications of aziridinium ions. Selective syntheses of alpha, beta-diamino esters,
alpha-sulfanyl-beta-amino esters, beta-lactams, and 1,5-benzodiazepin-2-one. Organic Letters. [IF=1.091, Cited=10, 11073643].
Petrassi HM, Sharpless KB, Kelly JW (2001) The copper-mediated cross-coupling of phenylboronic acids and
N-hydroxyphthalimide at room temperature: synthesis of aryloxyamines. Organic Letters. [IF=1.091, Cited=21, 11429858].
Demko ZP, Sharpless KB (2001) An intramolecular [2 + 3] cycloaddition route to fused 5-heterosubstituted tetrazoles.
Organic Letters. [IF=1.091, Cited=51, 11735592].
Demko ZP, Sharpless KB (2002) An expedient route to the tetrazole analogues of alpha-amino acids. Organic Letters.
[IF=1.091, Cited=34, 12123367].
Ripka AS, Díaz DD, Sharpless KB, Finn MG (2003) First practical synthesis of formamidine ureas and derivatives. Organic
Letters. [IF=1.091, Cited=2, 12713316].
Chan TR, Hilgraf R, Sharpless KB (2004) Polytriazoles as copper(I)-stabilizing ligands in catalysis. Organic Letters.
[IF=1.091, Cited=547, 15330631].
Krasiński A, Sharpless KB (2004) Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. Organic
Letters. [IF=1.091, Cited=64, 15070306].
Kalisiak J, Sharpless KB (2008) Efficient synthesis of 2-substituted-1,2,3-triazoles. Organic Letters. [IF=1.091,
Cited=44, 18597477].
Chuang TH, Sharpless KB (1999) Applications of aziridinium ions. Selective syntheses of beta-aryl-alpha,beta-diamino
esters. Organic Letters. [IF=1.091, Cited=6, 10825990].
Gontcharov AV, Liu H, Sharpless KB (1999) Tert-butylsulfonamide. A new nitrogen source for catalytic aminohydroxylation
and aziridination of olefins. Organic Letters. [IF=1.091, Cited=13, 10823205].
Gao B, Zhang L, Zheng Q, ..., Sharpless KB (2017) Bifluoride-catalysed sulfur(VI) fluoride exchange reaction for the
synthesis of polysulfates and polysulfonates. Nature Chemistry. [IF=3.667, Cited=70, 29064495].
Hong S, Shi Y, Wu NC, ..., Wu P (2019) Bacterial glycosyltransferase-mediated cell-surface chemoenzymatic glycan
modification. Nature Communications. [IF=3.268, Cited=20, 30996301].
Brighty GJ, Botham RC, Li S, ..., Kelly JW (2020) Using sulfuramidimidoyl fluorides that undergo sulfur(VI) fluoride
exchange for inverse drug discovery. Nature Chemistry. [IF=3.667, Cited=32, 32868886].
Li S, Li G, Gao B, ..., Sharpless KB (2021) SuFExable polymers with helical structures derived from thionyl
tetrafluoride. Nature Chemistry. [IF=3.667, Cited=25, 34400816].
Miyamoto Y, Kalisiak J, Korthals K, ..., Eckmann L (2013) Expanded therapeutic potential in activity space of next-
generation 5-nitroimidazole antimicrobials with broad structural diversity. Proceedings of the National Academy of
Sciences of the United States of America. [IF=2.765, Cited=34, 24101497].
Hirose T, Maita N, Gouda H, ..., Sunazuka T (2013) Observation of the controlled assembly of preclick components in the
in situ click chemistry generation of a chitinase inhibitor. Proceedings of the National Academy of Sciences of the
United States of America. [IF=2.765, Cited=11, 24043811].
Zheng Q, Woehl JL, Kitamura S, ..., Sharpless KB (2019) SuFEx-enabled, agnostic discovery of covalent inhibitors of
human neutrophil elastase. Proceedings of the National Academy of Sciences of the United States of America. [IF=2.765,
Cited=71, 31484779].
Zhang J, Zhao X, Cappiello JR, ..., Sharpless KB (2021) Identification of simple arylfluorosulfates as potent agents
against resistant bacteria. Proceedings of the National Academy of Sciences of the United States of America. [IF=2.765,
Cited=8, 34244433].
Cheng Y, Li G, Smedley CJ, ..., Sharpless KB (2022) Diversity oriented clicking delivers β-substituted alkenyl sulfonyl
fluorides as covalent human neutrophil elastase inhibitors. Proceedings of the National Academy of Sciences of the
United States of America. [IF=2.765, Cited=6, 36070343].
Xin Y, Liu S, Liu Y, ..., Shui W (2023) Affinity selection of double-click triazole libraries for rapid discovery of
allosteric modulators for GLP-1 receptor. Proceedings of the National Academy of Sciences of the United States of
America. [IF=2.765, Cited=2, 36893261].
Kitamura S, Lin TH, Lee CCD, ..., Wolan DW (2024) Ultrapotent influenza hemagglutinin fusion inhibitors developed
through SuFEx-enabled high-throughput medicinal chemistry. Proceedings of the National Academy of Sciences of the United
States of America. [IF=2.765, Cited=0, 38753503].
Taylor P, Shyong YJ, Samskey N, ..., Camacho-Hernandez GA (2021) Ligand design for human acetylcholinesterase and
nicotinic acetylcholine receptors, extending beyond the conventional and canonical. Journal of Neurochemistry.
[IF=1.089, Cited=3, 33638151].
Sit RK, Kovarik Z, Maček Hrvat N, ..., Taylor P (2018) Pharmacology, Pharmacokinetics, and Tissue Disposition of
Zwitterionic Hydroxyiminoacetamido Alkylamines as Reactivating Antidotes for Organophosphate Exposure. Journal of
Pharmacology and Experimental Therapeutics. [IF=0.906, Cited=16, 30190337].
Shyong YJ, Sepulveda Y, Garcia A, ..., Taylor P (2021) Enhancing Target Tissue Levels and Diminishing Plasma Clearance
of Ionizing Zwitterionic Antidotes in Organophosphate Exposures. Journal of Pharmacology and Experimental Therapeutics.
[IF=0.906, Cited=1, 34145064].
Vanacore R, Ham AJL, Voehler M, ..., Hudson BG (2009) A sulfilimine bond identified in collagen IV. Science. [IF=7.729,
Cited=125, 19729652].
Crispino GA, Ho PT, Sharpless KB (1993) Selective perhydroxylation of squalene: taming the arithmetic demon. Science.
[IF=7.729, Cited=12, 8418495].
Kim WJ, Korthals KA, Li S, ..., Eckmann L (2017) Click Chemistry-Facilitated Structural Diversification of
Nitrothiazoles, Nitrofurans, and Nitropyrroles Enhances Antimicrobial Activity against Giardia lamblia. Antimicrobial
Agents and Chemotherapy. [IF=1.175, Cited=2, 28396548].
Gastaminza P, Pitram SM, Dreux M, ..., Chisari FV (2011) Antiviral stilbene 1,2-diamines prevent initiation of hepatitis
C virus RNA replication at the outset of infection. Journal of Virology. [IF=1.075, Cited=6, 21430055].
Toguchi S, Hirose T, Yorita K, ..., Sunazuka T (2015) In Situ Click Chemistry for the Identification of a Potent D-Amino
Acid Oxidase Inhibitor. Chemical and Pharmaceutical Bulletin. [IF=0.569, Cited=3, 26686243].
Lauwaet T, Miyamoto Y, Ihara S, ..., Eckmann L (2020) Click chemistry-facilitated comprehensive identification of
proteins adducted by antimicrobial 5-nitroimidazoles for discovery of alternative drug targets against giardiasis. PLoS
Neglected Tropical Diseases. [IF=1.335, Cited=6, 32302296].
Sharpless KB, Manetsch R (2006) In situ click chemistry: a powerful means for lead discovery. Expert Opinion on Drug
Discovery. [IF=1.259, Cited=48, 23506064].
Sharpless KB (2002) Searching for new reactivity (Nobel lecture). Angewandte Chemie - International Edition. [IF=2.456,
Cited=44, 19746596].
Homer JA, Xu L, Kayambu N, ..., Moses JE (2023) Sulfur fluoride exchange. Nature Reviews Methods Primers. [IF=10.589,
Cited=2, 38873592].

Publication with MISSING institution:

Goossen LJ, Liu H, Dress KR, Sharpless KB (1999) Catalytic asymmetric aminohydroxylation with amino-substituted
heterocycles as nitrogen sources. Angewandte Chemie - International Edition. [IF=2.456, Cited=5, 25138500].
Kolb HC, Finn MG, Sharpless KB (2001) Click Chemistry: Diverse Chemical Function from a Few Good Reactions. Angewandte
Chemie - International Edition. [IF=2.456, Cited=1000, 11433435].
Fokin VV, Sharpless KB (2001) A Practical and Highly Efficient Aminohydroxylation of Unsaturated Carboxylic Acids We
thank the National Institute of General Medical Sciences, the National Institutes of Health (GM 28384), National Science
Foundation (CHE-9985553), and the W. M. Keck Foundation for financial support. We are also grateful to Prof. M. G. Finn,
Dr. Wallace Pringle, and Dr. A. Erik Rubin for many helpful discussions. Angewandte Chemie - International Edition.
[IF=2.456, Cited=7, 11592169].
Andersson MA, Epple R, Sharpless KB (2002) A new approach to osmium-catalyzed asymmetric dihydroxylation and
aminohydroxylation of olefins. Angewandte Chemie - International Edition. [IF=2.456, Cited=17, 12491382].
Lewis WG, Green LG, Grynszpan F, ..., Sharpless KB (2002) Click chemistry in situ: acetylcholinesterase as a reaction
vessel for the selective assembly of a femtomolar inhibitor from an array of building blocks. Angewandte Chemie -
International Edition. [IF=2.456, Cited=229, 12491310].
Rostovtsev VV, Green LG, Sharpless KB (2002) A stepwise huisgen cycloaddition process: copper(I)-catalyzed
regioselective "ligation" of azides and terminal alkynes. Angewandte Chemie - International Edition. [IF=2.456,
Cited=1000, 12203546].
Wu P, Feldman AK, Nugent AK, ..., Sharpless KB (2004) Efficiency and fidelity in a click-chemistry route to triazole
dendrimers by the copper(i)-catalyzed ligation of azides and alkynes. Angewandte Chemie - International Edition.
[IF=2.456, Cited=211, 15274216].
Mocharla VP, Colasson B, Lee LV, ..., Wong CH (2004) In situ click chemistry: enzyme-generated inhibitors of carbonic
anhydrase II. Angewandte Chemie - International Edition. [IF=2.456, Cited=72, 15599912].
Narayan S, Muldoon J, Finn MG, Sharpless KB (2005) "On water": unique reactivity of organic compounds in aqueous
suspension. Angewandte Chemie - International Edition. [IF=2.456, Cited=271, 15844112].
Whiting M, Muldoon J, Lin YC, ..., Elder JH (2006) Inhibitors of HIV-1 protease by using in situ click chemistry.
Angewandte Chemie - International Edition. [IF=2.456, Cited=136, 16425339].
Yoo EJ, Ahlquist M, Kim SH, ..., Chang S (2007) Copper-catalyzed synthesis of N-sulfonyl-1,2,3-triazoles: controlling
selectivity. Angewandte Chemie - International Edition. [IF=2.456, Cited=59, 17397087].
Agnew HD, Rohde RD, Millward SW, ..., Sharpless KB (2009) Iterative in situ click chemistry creates antibody-like
protein-capture agents. Angewandte Chemie - International Edition. [IF=2.456, Cited=49, 19301344].
Hein JE, Tripp JC, Krasnova LB, Sharpless KB (2009) Copper(I)-catalyzed cycloaddition of organic azides and
1-iodoalkynes. Angewandte Chemie - International Edition. [IF=2.456, Cited=89, 19774581].
Dong J, Krasnova L, Finn MG, Sharpless KB (2014) Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click
chemistry. Angewandte Chemie - International Edition. [IF=2.456, Cited=259, 25112519].
Minond D, Saldanha SA, Subramaniam P, ..., Hodder P (2009) Inhibitors of VIM-2 by screening pharmacologically active and
click-chemistry compound libraries. Bioorganic and Medicinal Chemistry. [IF=0.86, Cited=25, 19553129].
Sugawara A, Sunazuka T, Hirose T, ..., Omura S (2007) Design and synthesis via click chemistry of
8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity. Bioorganic and Medicinal Chemistry
Letters. [IF=0.704, Cited=6, 17869508].
Bourne Y, Radić Z, Sharpless KB, ..., Marchot P (2005) Structural insights into conformational flexibility at the
peripheral site and within the active center gorge of AChE. Chemico-Biological Interactions. [IF=1.057, Cited=9, 16259971].
Radić Z, Manetsch R, Krasiński A, ..., Taylor P (2005) Molecular basis of interactions of cholinesterases with tight
binding inhibitors. Chemico-Biological Interactions. [IF=1.057, Cited=11, 16289416].
Radić Z, Manetsch R, Fournier D, ..., Taylor P (2008) Probing gorge dimensions of cholinesterases by freeze-frame click
chemistry. Chemico-Biological Interactions. [IF=1.057, Cited=2, 18555981].
Radić Z, Kalisiak J, Sharpless KB, Taylor P (2010) Interaction kinetics of oximes with native, phosphylated and aged
human acetylcholinesterase. None. [IF=None, Cited=9, 20412789].
Sharpless KB (2003) The growing impact of click chemistry on drug discovery. Drug Discovery Today. [IF=1.663,
Cited=1000, 14678739].
Elbein AD, Szumilo T, Sanford BA, ..., Adams C (1987) Effect of isomers of swainsonine on glycosidase activity and
glycoprotein processing. Biochemistry. [IF=0.753, Cited=9, 3111529].
Sharpless KB, Flood TC (1971) Oxotransition metal oxidants as mimics for the action of mixed-function oxygenases. "NIH
shift" with chromyl reagents. Journal of the American Chemical Society. [IF=2.573, Cited=9, 5553075].
Tanaka S, Yamamoto H, Nozaki H, ..., Cutting JD (1974) Stereoselective epoxidations of acyclic allylic alcohols by
transition metal--hydroperoxide reagents. Synthesis of dl-C18 Cecropia juvenile hormone from farnesol. Journal of the
American Chemical Society. [IF=2.573, Cited=11, 4854400].
van Tamelen EE, Sharpless KB, Hanzlik R, ..., Wszolek PC (1967) Enzymic cyclization of
trans,trans,trans-18,19-dihydrosqualene 2,3-oxide. Journal of the American Chemical Society. [IF=2.573, Cited=5, 6064361].
Sharpless KB, Snyder TE, Spencer TA, ..., Nelson JA (1969) Biological demethylation of 4,4-dimethyl sterols, Evidence
for enzymic epimerization of the 4beta-methyl group prior to its oxidative removal. Journal of the American Chemical
Society. [IF=2.573, Cited=5, 5791927].
Kitamura S, Zheng Q, Woehl JL, ..., Wolan DW (2020) Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput
Medicinal Chemistry. Journal of the American Chemical Society. [IF=2.573, Cited=43, 32479075].
Hirose T, Sunazuka T, Sugawara A, ..., Omura S (2009) Chitinase inhibitors: extraction of the active framework from
natural argifin and use of in situ click chemistry. Journal of Antibiotics. [IF=0.805, Cited=22, 19329983].
Wu P, Malkoch M, Hunt JN, ..., Hawker CJ (2005) Multivalent, bifunctional dendrimers prepared by click chemistry.
Chemical Communications. [IF=0.902, Cited=86, 16307142].
Sit RK, Radić Z, Gerardi V, ..., Taylor P (2011) New structural scaffolds for centrally acting oxime reactivators of
phosphylated cholinesterases. Journal of Biological Chemistry. [IF=1.122, Cited=65, 21464125].
Cochran R, Kalisiak J, Küçükkilinç T, ..., Taylor P (2011) Oxime-assisted acetylcholinesterase catalytic scavengers of
organophosphates that resist aging. Journal of Biological Chemistry. [IF=1.122, Cited=26, 21730071].
Radić Z, Sit RK, Kovarik Z, ..., Taylor P (2012) Refinement of structural leads for centrally acting oxime reactivators
of phosphylated cholinesterases. Journal of Biological Chemistry. [IF=1.122, Cited=55, 22343626].
Yamauchi JG, Gomez K, Grimster N, ..., Taylor P (2012) Synthesis of selective agonists for the α7 nicotinic
acetylcholine receptor with in situ click-chemistry on acetylcholine-binding protein templates. Molecular Pharmacology.
[IF=0.939, Cited=7, 22784805].
Kalantar TH, Sharpless KB (1993) Transformations of hydroxy cyclic sulfates: stereospecific conversion into
2,3,5-trisubstituted tetrahydrofurans. None. [IF=None, Cited=0, 8435231].
Li G, Sharpless KB (1996) Catalytic asymmetric aminohydroxylation provides a short taxol side-chain synthesis. None.
[IF=None, Cited=8, 8756354].
Kwok SW, Hein JE, Sharpless KB (2008) REGIOSELECTIVE SYNTHESIS OF EITHER 1H- OR 2H-1,2,3- TRIAZOLES VIA MICHAEL ADDITION
TO α,ß-UNSATURATED KETONES. Heterocycles. [IF=0.215, Cited=4, 19802363].
Demko ZP, Sharpless KB (2002) A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis
of 5-sulfonyl tetrazoles from azides and sulfonyl cyanides. Angewandte Chemie - International Edition. [IF=2.456,
Cited=25, 19746612].
Demko ZP, Sharpless KB (2002) A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis
of 5-acyltetrazoles from azides and acyl cyanides. Angewandte Chemie - International Edition. [IF=2.456, Cited=23, 19746613].
Rahman R, Sharpless KB, Spencer TA, Clayton RB (1970) Removal of the 4,4-dimethyl carbons in the enzymic conversion of
lanosterol to cholesterol. Initial loss of the 4-alpha-methyl group. Journal of Biological Chemistry. [IF=1.122,
Cited=13, 5445804].
Willett JD, Sharpless KB, Lord KE, ..., Clayton RB (1967) Squalene-2,3oxide, an intermediate in the enzymatic conversion
of squalene to lanosterol and cholesterol. Journal of Biological Chemistry. [IF=1.122, Cited=32, 6061706].

Sharpless, K Barry

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