Krska, Shane

Publication with MATCHING institution:

Chen X, Wei Z, Huang KH, ..., Cooks RG (2022) Pd Reaction Intermediates in Suzuki-Miyaura Cross-Coupling Characterized
by Mass Spectrometry. ChemPlusChem. [IF=0.703, Cited=1, 35112808].
Liu K, Kurukulasuriya R, Dykstra K, ..., Cernak T (2019) Development of indazole mineralocorticoid receptor antagonists
and investigation into their selective late-stage functionalization. Bioorganic and Medicinal Chemistry Letters.
[IF=0.704, Cited=0, 31104995].
Golden DL, Flynn KM, Aikonen S, ..., Stahl SS (2024) Radical Chlorination of Non-Resonant Heterobenzylic C-H Bonds and
High-Throughput Diversification of Heterocycles. Chem. [IF=2.863, Cited=0, 39108591].
Wleklinski M, Carpenter PM, Dykstra KD, ..., Ferguson RD (2024) Parallel purification of microscale libraries via
automated solid phase extraction. SLAS Technology. [IF=0.671, Cited=0, 38423211].
Dreher SD, Krska S (2021) Chemistry Informer Libraries: Conception, Early Experience, and Role in the Future of
Cheminformatics. Accounts of Chemical Research. [IF=3.533, Cited=15, 33723992].
Chen SJ, Krska S, Krska SW, ..., Stahl SS (2023) Copper-Catalyzed Benzylic C-H Cross-Coupling Enabled by Redox Buffers:
Expanding Synthetic Access to Three-Dimensional Chemical Space. Accounts of Chemical Research. [IF=3.533, Cited=1, 38051914].
Cao W, Maza JC, Chernyak N, ..., Francis MB (2023) Modification of Cysteine-Substituted Antibodies Using Enzymatic
Oxidative Coupling Reactions. Bioconjugate Chemistry. [IF=0.921, Cited=3, 36787347].
Boga SB, Krska S, Lin S, ..., Parish CA (2019) Site-Selective Synthesis of Insulin Azides and Bioconjugates.
Bioconjugate Chemistry. [IF=0.921, Cited=1, 30946565].
Tyagarajan S, Lowden CT, Peng Z, ..., Krska S (2015) Heterocyclic Regioisomer Enumeration (HREMS): A Cheminformatics
Design Tool. Journal of Chemical Information and Modeling. [IF=1.379, Cited=2, 26017267].
Chinn AJ, Hwang J, Kim B, ..., Miller SJ (2020) Application of High-Throughput Competition Experiments in the
Development of Aspartate-Directed Site-Selective Modification of Tyrosine Residues in Peptides. Journal of Organic
Chemistry. [IF=0.885, Cited=1, 32614587].
King RP, Krska S, Buchwald SL (2021) A Ligand Exchange Process for the Diversification of Palladium Oxidative Addition
Complexes. Organic Letters. [IF=1.091, Cited=1, 34319123].
King RP, Krska S, Buchwald SL (2021) A Neophyl Palladacycle as an Air- and Thermally Stable Precursor to Oxidative
Addition Complexes. Organic Letters. [IF=1.091, Cited=1, 34613744].
Dykstra KD, Streckfuss E, Liu M, ..., Krska S (2021) Synthesis of HDAC Inhibitor Libraries via Microscale Workflow. ACS
Medicinal Chemistry Letters. [IF=0.873, Cited=3, 33738059].
Ichiishi N, Moore KP, Wassermann AM, ..., Krska S (2018) Reducing Limitation in Probe Design: The Development of a
Diazirine-Compatible Suzuki-Miyaura Cross Coupling Reaction. ACS Medicinal Chemistry Letters. [IF=0.873, Cited=4, 30655947].
Chen SJ, Golden DL, Krska S, ..., Stahl SS (2021) Copper-Catalyzed Cross-Coupling of Benzylic C-H Bonds and Azoles with
Controlled N-Site Selectivity. Journal of the American Chemical Society. [IF=2.573, Cited=15, 34464528].
Maity S, Lopez MA, Bates DM, ..., Stahl SS (2023) Polar Heterobenzylic C(sp³)-H Chlorination Pathway Enabling
Efficient Diversification of Aromatic Nitrogen Heterocycles. Journal of the American Chemical Society. [IF=2.573,
Cited=1, 37642292].
Maza JC, Bader DLV, Xiao L, ..., Francis MB (2019) Enzymatic Modification of N-Terminal Proline Residues Using Phenol
Derivatives. Journal of the American Chemical Society. [IF=2.573, Cited=17, 30726077].
Maligres PE, Krska S, Dormer PG (2012) A soluble copper(I) source and stable salts of volatile ligands for copper-
catalyzed C-X couplings. Journal of Organic Chemistry. [IF=0.885, Cited=1, 22881453].
Limanto J, Shultz CS, Dorner B, ..., Krska S (2008) Synthesis of a tertiary carbinamide via a novel Rh-catalyzed
asymmetric hydrogenation. Journal of Organic Chemistry. [IF=0.885, Cited=5, 18186647].
Maligres PE, Krska S, Humphrey GR (2004) Enantioselective hydrogenation of alpha-aryloxy alpha,beta-unsaturated acids.
Asymmetric synthesis of alpha-aryloxycarboxylic acids. Organic Letters. [IF=1.091, Cited=4, 15330609].
Krska S, Alorati A, Baxter JM, ..., Davies IW (2010) Asymmetric hydrogenation of protected allylic amines. Organic
Letters. [IF=1.091, Cited=9, 20735080].
Hu H, Chen SJ, Mandal M, ..., Stahl SS (2020) Copper-catalysed benzylic C-H coupling with alcohols via radical relay
enabled by redox buffering. Nature Catalysis. [IF=5.117, Cited=35, 32368720].
Chen SJ, He CQ, Kong M, ..., Stahl SS (2023) Accessing three-dimensional molecular diversity through benzylic C-H cross-
coupling. None. [IF=None, Cited=1, 38463240].
Maza JC, Ramsey AV, Mehare M, ..., Francis MB (2020) Secondary modification of oxidatively-modified proline N-termini
for the construction of complex bioconjugates. Organic and Biomolecular Chemistry. [IF=0.77, Cited=5, 32100807].
Suh SE, Nkulu LE, Lin S, ..., Stahl SS (2021) Benzylic C-H isocyanation/amine coupling sequence enabling high-throughput
synthesis of pharmaceutically relevant ureas. Chemical Science. [IF=1.563, Cited=10, 34377424].
Chambers RK, Weaver JD, Kim J, ..., White MC (2023) A preparative small-molecule mimic of liver CYP450 enzymes in the
aliphatic C-H oxidation of carbocyclic N-heterocycles. Proceedings of the National Academy of Sciences of the
United States of America. [IF=2.765, Cited=3, 37428920].
Uehling MR, King RP, Krska S, ..., Buchwald SL (2019) Pharmaceutical diversification via palladium oxidative addition
complexes. Science. [IF=7.729, Cited=43, 30679373].
Vasilopoulos A, Krska S, Krska SW, ..., Stahl SS (2021) C(sp³)-H methylation enabled by peroxide
photosensitization and Ni-mediated radical coupling. Science. [IF=7.729, Cited=35, 33888639].
Prieto Kullmer CN, Kautzky JA, Krska S, ..., MacMillan DWC (2022) Accelerating reaction generality and mechanistic
insight through additive mapping. Science. [IF=7.729, Cited=26, 35482871].

Publication with MISMATCHING institution:

Cohen RD, Saurí J, Huff CA, ..., Martin GE (2016) Additional pitfalls of using 1,1-ADEQUATE for structure elucidation.
Magnetic Resonance in Chemistry. [IF=0.681, Cited=4, 27396947].
Krska S, DiRocco DA, Dreher SD, Shevlin M (2017) The Evolution of Chemical High-Throughput Experimentation To Address
Challenging Problems in Pharmaceutical Synthesis. Accounts of Chemical Research. [IF=3.533, Cited=71, 29172435].
Huff CA, Cohen RD, Dykstra KD, ..., Krska S (2016) Photoredox-Catalyzed Hydroxymethylation of Heteroaromatic Bases.
Journal of Organic Chemistry. [IF=0.885, Cited=24, 27315015].
Shen F, Tyagarajan S, Perera D, ..., Maleczka RE (2016) Bismuth Acetate as a Catalyst for the Sequential
Protodeboronation of Di- and Triborylated Indoles. Organic Letters. [IF=1.091, Cited=11, 26998615].
McCammant MS, Thompson S, Brooks AF, ..., Sanford MS (2017) Cu-Mediated C-H ¹⁸F-Fluorination of Electron-Rich
(Hetero)arenes. Organic Letters. [IF=1.091, Cited=29, 28665619].
Shultz CS, Krska S (2007) Unlocking the potential of asymmetric hydrogenation at Merck. Accounts of Chemical Research.
[IF=3.533, Cited=36, 18020425].
Krska S, Hughes DL, Reamer RA, ..., Trost BM (2002) The unusual role of CO transfer in molybdenum-catalyzed asymmetric
alkylations. Journal of the American Chemical Society. [IF=2.573, Cited=8, 12392401].
Lloyd-Jones G, Lloyd-Jones GC, Krska S, ..., Reamer RA (2004) Conclusive evidence for a retention-retention pathway for
the molybdenum-catalyzed asymmetric alkylation. Journal of the American Chemical Society. [IF=2.573, Cited=16, 14733529].
Hsiao Y, Rivera NR, Rosner T, ..., Malan C (2004) Highly efficient synthesis of beta-amino acid derivatives via
asymmetric hydrogenation of unprotected enamines. Journal of the American Chemical Society. [IF=2.573, Cited=49, 15303855].
Strotman NA, Baxter CA, Brands KMJ, ..., Wright TJ (2011) Reaction development and mechanistic study of a ruthenium
catalyzed intramolecular asymmetric reductive amination en route to the dual Orexin inhibitor Suvorexant (MK-4305).
Journal of the American Chemical Society. [IF=2.573, Cited=23, 21528938].
Schmink JR, Krska S (2011) Reversed-polarity synthesis of diaryl ketones via palladium-catalyzed cross-coupling of
acylsilanes. Journal of the American Chemical Society. [IF=2.573, Cited=20, 22070616].
Preshlock SM, Ghaffari B, Maligres PE, ..., Smith MR (2013) High-throughput optimization of Ir-catalyzed C-H borylation:
a tutorial for practical applications. Journal of the American Chemical Society. [IF=2.573, Cited=54, 23534698].
Ghaffari B, Preshlock SM, Plattner DL, ..., Smith MR (2014) Silyl phosphorus and nitrogen donor chelates for homogeneous
ortho borylation catalysis. Journal of the American Chemical Society. [IF=2.573, Cited=32, 25141136].
Hansen KB, Hsiao Y, Xu F, ..., Armstrong JD (2009) Highly efficient asymmetric synthesis of sitagliptin. Journal of the
American Chemical Society. [IF=2.573, Cited=55, 19507853].
Zuckerman RL, Krska SW, Krska S, ..., Bergman RG (2000) Zirconium-mediated metathesis of imines: a study of the scope,
longevity, and mechanism of a complicated catalytic system. Journal of the American Chemical Society. [IF=2.573,
Cited=29, 16636698].
Webb EW, Cheng K, Winton WP, ..., Scott PJH (2024) Development of High-Throughput Experimentation Approaches for Rapid
Radiochemical Exploration. Journal of the American Chemical Society. [IF=2.573, Cited=0, 38580459].
Molinaro C, Shultz S, Roy A, ..., Krska S (2011) A practical synthesis of renin inhibitor MK-1597 (ACT-178882) via
catalytic enantioselective hydrogenation and epimerization of piperidine intermediate. Journal of Organic Chemistry.
[IF=0.885, Cited=1, 21250716].
Zhong YL, Gauthier DR, Shi YJ, ..., Yasuda N (2012) Synthesis of antifungal glucan synthase inhibitors from
enfumafungin. Journal of Organic Chemistry. [IF=0.885, Cited=3, 22423625].
Chobanian HR, Guo Y, Liu P, ..., DeVita RJ (2014) Discovery of MK-4409, a Novel Oxazole FAAH Inhibitor for the Treatment
of Inflammatory and Neuropathic Pain. ACS Medicinal Chemistry Letters. [IF=0.873, Cited=7, 24944750].
Shultz CS, Dreher SD, Ikemoto N, ..., Dimichele L (2005) Asymmetric hydrogenation of N-sulfonylated-alpha-dehydroamino
acids: toward the synthesis of an anthrax lethal factor inhibitor. Organic Letters. [IF=1.091, Cited=14, 16048303].
Mangion IK, Chen Cy, Li H, ..., Zavialov I (2014) Enantioselective synthesis of an HCV NS5a antagonist. Organic Letters.
[IF=1.091, Cited=9, 24724971].
Zhong YL, Krska S, Zhou H, ..., Askin D (2009) Catalytic asymmetric synthesis of an HIV integrase inhibitor. Organic
Letters. [IF=1.091, Cited=8, 19099496].
Limanto J, Krska S, Dorner BT, ..., Tan L (2010) Dynamic kinetic resolution: asymmetric transfer hydrogenation of alpha-
alkyl-substituted beta-ketoamides. Organic Letters. [IF=1.091, Cited=15, 20028132].
Cernak T, Dykstra KD, Tyagarajan S, ..., Krska S (2015) The medicinal chemist's toolbox for late stage functionalization
of drug-like molecules. Chemical Society Reviews. [IF=8.116, Cited=404, 26507237].
Kutchukian PS, Dropinski JF, Dykstra KD, ..., Dreher SD (2016) Chemistry informer libraries: a chemoinformatics enabled
approach to evaluate and advance synthetic methods. Chemical Science. [IF=1.563, Cited=75, 28660032].
Cernak T, Dykstra KD, Tyagarajan S, ..., Krska S (2017) Correction: The medicinal chemist's toolbox for late stage
functionalization of drug-like molecules. Chemical Society Reviews. [IF=8.116, Cited=0, 28280821].
Liu W, Huang X, Placzek MS, ..., Groves JT (2017) Site-selective ¹⁸F fluorination of unactivated C-H bonds
mediated by a manganese porphyrin. Chemical Science. [IF=1.563, Cited=25, 29675161].
Ichiishi N, Caldwell JP, Lin M, ..., Krska S (2018) Protecting group free radical C-H trifluoromethylation of peptides.
Chemical Science. [IF=1.563, Cited=38, 29780547].
Hughes DL, Lloyd-Jones G, Lloyd-Jones GC, ..., Reamer RA (2004) Mechanistic studies of the molybdenum-catalyzed
asymmetric alkylation reaction. Proceedings of the National Academy of Sciences of the United States of America.
[IF=2.765, Cited=6, 15056759].
Friedfeld MR, Shevlin M, Hoyt JM, ..., Chirik PJ (2013) Cobalt precursors for high-throughput discovery of base metal
asymmetric alkene hydrogenation catalysts. Science. [IF=7.729, Cited=86, 24288328].

Publication with MISSING institution:

Ruck RT, Krska S, Krska SW, Bergman RG (2004) Carboamination: additions of imine C=N bonds across alkynes catalyzed by
imidozirconium complexes. Angewandte Chemie - International Edition. [IF=2.456, Cited=16, 15468090].
Maligres PE, Li J, Krska S, ..., Raheem IT (2012) C-O cross-coupling of activated aryl and heteroaryl halides with
aliphatic alcohols. Angewandte Chemie - International Edition. [IF=2.456, Cited=14, 22887962].
Preshlock SM, Plattner DL, Maligres PE, ..., Smith MR (2013) A traceless directing group for C-H borylation. Angewandte
Chemie - International Edition. [IF=2.456, Cited=41, 24222178].
Dirocco DA, Dykstra K, Krska S, ..., Tudge M (2014) Late-stage functionalization of biologically active heterocycles
through photoredox catalysis. Angewandte Chemie - International Edition. [IF=2.456, Cited=119, 24677697].
Chang M, Huang Y, Liu S, ..., Zhang X (2014) Asymmetric hydrogenation of pyridinium salts with an iridium phosphole
catalyst. Angewandte Chemie - International Edition. [IF=2.456, Cited=26, 25297378].
Hansen KB, Hsiao Y, Xu F, ..., Armstrong JD (2020) Correction to "Highly Efficient Asymmetric Synthesis of Sitagliptin".
Journal of the American Chemical Society. [IF=2.573, Cited=0, 32706576].
Iida T, Satoh H, Maeda K, ..., Volante RP (2005) Practical synthesis of a neuropeptide Y antagonist via stereoselective
addition to a ketene. Journal of Organic Chemistry. [IF=0.885, Cited=3, 16268594].
Trost BM, Dogra K, Hachiya I, ..., Reider PJ (2002) Designed ligands as probes for the catalytic binding mode in Mo-
catalyzed asymmetric allylic alkylation. Angewandte Chemie - International Edition. [IF=2.456, Cited=0, 19750636].